種別 タイトル 著者 誌名 巻号 ページ 出版年 DOI URL 原著論文 "Ex vivo imaging and analysis of ROS generation correlated with microglial activation in rat model with acute neuroinflammation induced by intrastriatal injection of LPS." "M. Shukuri, M. Uchino, T. Sakamaki, S. Onoe, R. Hosoi, K. Todoroki, Y. Arano, T. Sakai, H. Akizawa, O. Inoue." "Biochem. Biophys. Res. Commun." 584 101-106 2021 原著論文 "Influence of linker molecules in hexavalent RGD peptides on their multivalent interactions with integrin αvβ3." "Y. Mizuno, K. Kimura, S. Onoe, M. Shukuri, Y. Kuge, H. Akizawa." "J. Med. Chem." 64(21) 16008-16019 2021 原著論文 "Aryl isocyanide derivative for one-pot synthesis of purification-free 99mTc-labeled hexavalent targeting probe." "Y. Mizuno, T. Uehara, C. Jen, H. Akizawa, Y. Arano." "Nucl. Med. Biol." 86-87 30-36 2020 原著論文 "The synthesis of a 99mTc-labeled tetravalent targeting probe upon isonitrile coordination to 99mTcI for enhanced target uptake in saturable systems." "Y. Mizuno, T. Uehara, C. Jen, H. Akizawa, Y. Arano." "RSC Adv." 9 26126-26135 2019 原著論文 "Coordination-mediated synthesis of purification-free bivalent 99mTc-labeled probes for in vivo imaging of saturable system." "Y. Taira, T. Uehara, M. Tsuchiya, H. Takemori, Y. Mizuno, S. Takahashi, H. Suzuki, H. Hanaoka, H. Akizawa, Y. Arano." "Bioconjugate Chem." 29(2) 459-466 2018 原著論文 "111In-DTPA-D-Phe-1-Asp0-D-Phe1-octreotide exhibits higher tumor accumulation and lower renal radioactivity than 111In-DTPA-D-Phe1-octreotide." "N. Oshima, H. Akizawa, H. Kitaura, H. Kawashima, S. Zhao, Y. Zhao, K. Nishijima, Y. Kitamura, Y. Arano, Y. Kuge, K. Ohkura." "Nucl. Med. Biol." 54 18-26 2017 原著論文 "Redesign of negatively charged 111In-DTPA-octreotide derivative to reduce renal radioactivity." "N. Oshima, H. Akizawa, H. Kawashima, S. Zhao, Y. Zhao, K. Nishijima, Y. Kitamura, Y. Arano, Y. Kuge, K. Ohkura." "Nucl. Med. Biol." 48 16-25 2017 原著論文 "The Thymidine Phosphorylase Imaging Agent 123I-IIMU Predicts the Efficacy of Capecitabine." " N. Kobashi, H. Matsumoto, S. Zhao, S. Meike, Y. Okumura, T. Abe, H. Akizawa, K. Ohkura, K. Nishijima, N. Tamaki, Y. Kuge." "J. Nucl. Med." 57(8) 1276-1281 2016 原著論文 "Relationship between biodistribution of a novel thymidine phosphorylase (TP) imaging probe and TP expression levels in normal mice." "Zhao S, Li H, Nishijima K, Zhao Y, Akizawa H, Shimizu Y, Ohkura K, Tamaki N, Kuge Y." "Ann. Nucl. Med." 29(7) 582-587 2015 原著論文 "Design, synthesis and biological evaluation of negatively charged 111In-DTPA-octreotide derivatives." "N. Oshima, H. Akizawa, S. Zhao, Y. Zhao, K. Nishijima, Y. Kitamura, Y. Arano, Y. Kuge, K. Ohkura" "Bioorg. Med. Chem." 22(4) 1377-1382 2014 原著論文 "Renal brush border enzyme-cleavable linkages for low renal radioactivity levels of radiolabeled antibody fragments." "H. Akizawa, M. Imajima, H. Hanaoka, T. Uehara, S. Satake, Y. Arano." "Bioconjugate Chem." 24(2) 291-299 2013 原著論文 "Chemical Design of 99mTc-Labeled Probes for Targeting Osteogenic Bone Region." "M. Yanagi, T. Uehara, Y. Uchida, S. Kiyota, M. Kinoshita, Y. Higaki, H. Akizawa, H. Hanaoka, Y. Arano." "Bioconjugate Chem." 24(7) 1248-1255 2013 原著論文 "Versatile photorearrangement of photocycloadducts from 5-fluoro-1,3-dimethyluracil and naphthalene." "K. Ohkura, H. Akizawa, M. Kudo, T. Ishihara, N. Oshima, K. Seki." Heterocycles 84(2) 1057-1065 2012 原著論文 "Synthesis and evaluation of diastereoisomers of 1,4,7-triazacyclononane-1,4,7-tris-(glutaric acid) (NOTGA) for multimeric radiopharmaceuticals of gallium." "F. L. Guerra Gomez, T. Uehara, T. Rokugawa, Y. Higaki, H. Suzuki, H. Hanaoka, H. Akizawa, Y. Arano." "Bioconjugate Chem." 23(11) 2229-2238 2012 原著論文 "Radiolabeled uracil derivative as a novel SPECT probe for thymidine phosphorylase: Suppressed accumulation into tumor cells by target gene knockdown." "H. Li, S. Zhao, Y. Jin, K. Nishijima, H. Akizawa, K. Ohkura, N. Tamaki, Y. Kuge." "Nucl. Med. Commun." 32(12) 1211-1215 2011 原著論文 "Toward in vivo imaging of heart disease using a radiolabeled single-chain Fv fragment targeting tenascin-C." "N. Kobayashi, K. Odaka, T. Uehara, K. Imanaka-Yoshida, Y. Kato, H. Oyama, H. Tadokoro, H. Akizawa, S. Tanada, M. Hiroe, T. Fukumura, I. Komuro, Y. Arano, T. Yoshida, T. Irie." "Anal. Chem." 83(23) 9123-9130 2011