種別 タイトル 著者 誌名 巻号 ページ 出版年 DOI URL 原著論文 "Screening for Protein Kinase C Ligands Using Fluorescence Resonance Energy Transfer." "Nami Ohashi, Wataru Nomura*, Natsuki Minato & Hirokazu Tamamura*" "Chem. Pharm. Bull. (Tokyo)." 62 1019-1025 2014 10.1248/cpb.c14-00419 原著論文 "Isostere-based Design of 8-Azacoumarin-type Photolabile Protecting Groups: a Hydrophilicity-increasing Strategy for Coumarin-4-ylmethyls." "Tetsuo Narumi, Hikaru Takano, Nami Ohashi, Akinobu Suzuki, Toshiaki Furuta & Hirokazu Tamamura*" "Org. Lett." 16 1184-1187 2014 10.1021/ol5000583 原著論文 "A CD4 mimic as an HIV entry inhibitor: Pharmacokinetics." "Chie Hashimoto, Tetsuo Narumi, Hiroyuki Otsuki, Yuki Hirota, Hiroshi Arai, Kazuhisa Yoshimura, Shigeyoshi Harada, Nami Ohashi, Wataru Nomura, Tomoyuki Miura, Tatsuhiko Igarashi, Shuzo Matsushita & Hirokazu Tamamura*" "Bioorg. Med. Chem." 21 7884-7889 2013 10.1016/j.bmc.2013.10.005 原著論文 "Cell-Permeable Stapled Peptides Based on HIV-1 Integrase Inhibitors Derived from HIV-1 Gene Products." "Wataru Nomura, Haruo Aikawa, Nami Ohashi, Emiko Urano, Mathieu Métifiot, Masayuki Fujino, Kasthuraiah Maddali, Taro Ozaki, Ami Nozue, Tetsuo Narumi, Chie Hashimoto, Tomohiro Tanaka, Yves Pommier, Naoki Yamamoto, Jun A. Komano, Tsutomu Murakami & Hirokazu Tamamura*" "ACS Chem. Biol." 8 " 2235–2244" 2013 10.1021/cb400495h 原著論文 "CD4 Mimics as HIV Entry Inhibitors: Lead Optimization Studies of the Aromatic Substituents." "Tetsuo Narumi, Hiroshi Arai, Kazuhisa Yoshimura, Shigeyoshi Harada, Yuki Hirota, Nami Ohashi, Chie Hashimoto, Wataru Nomura, Shuzo Matsushita & Hirokazu Tamamura*" "Bioorg. Med. Chem." 21 "2518-2526 " 2013 10.1016/j.bmc.2013.02.041 原著論文 "Low-Molecular-Weight CXCR4 Ligands with Variable Spacers." "Tetsuo Narumi, Haruo Aikawa, Tomohiro Tanaka, Chie Hashimoto, Nami Ohashi, Wataru Nomura, Takuya Kobayakawa, Hikaru Takano, Yuki Hirota, Tsutomu Murakami, Naoki Yamamoto & Hirokazu Tamamura*" ChemMedChem " 8" 118-124 2013 10.1002/cmdc.201200390 原著論文 "Fluorescent-Responsive Synthetic C1b Domains of Protein Kinase C as Reporters of Specific High-Affinity Ligand Binding." "Nami Ohashi, Wataru Nomura*, Tetsuo Narumi, Nancy E. Lewin, Kyoko Itotani, Peter M. Blumberg & Hirokazu Tamamura*" "Bioconjugate Chem." 22 82-87 2012 10.1021/bc100414a 原著論文 "Fluorescence-Quenching Screening of Protein Kinase C Ligands with an Environmentally Sensitive Fluorophore." "Wataru Nomura, Nami Ohashi, Yoshiaki Okuda, Tetsuo Narumi, Teikichi Ikura, Nobutoshi Ito & Hirokazu Tamamura*" "Bioconjugate Chem." 22 923-930 2011 10.1021/bc100567k 原著論文 "Synthetic Caged DAG-lactones for Photochemically Controlled Activation of Protein Kinase C." "Wataru Nomura, Tetsuo Narumi, Nami Ohashi, Yuki Serizawa, Nancy E. Lewin, Peter M. Blumberg, Toshiaki Furuta & Hirokazu Tamamura*" ChemBioChem 12 535-539 2011 10.1002/cbic.201000670 原著論文 "Azamacrocyclic Metal Complexes as CXCR4 Antagonists." "Tomohiro Tanaka, Tetsuo Narumi*, Taro Ozaki, Akira Sohma, Nami Ohashi, Chie Hashimoto, Kyoko Itotani, Wataru Nomura, Tsutomu Murakami, Naoki Yamamoto & Hirokazu Tamamura*" ChemMedChem 6 834-839 2011 10.1002/cmdc.201000548 原著論文 "CD4 Mimics Targeting the HIV Entry Mmechanism and Their Hybrid Molecules." "Tetsuo Narumi, Chihiro Ochiai, Kazuhisa Yoshimura, Shigeyoshi Harada, Tomohiro Tanaka, Wataru Nomura, Hiroshi Arai, Taro Ozaki, Nami Ohashi, Matsushita Shuzo & Hirakazu Tamamura*" "Bioorg. Med. Chem. Lett." 20 5853-5858 2010 10.1016/j.bmcl.2010.07.106 原著論文 "Peptidic HIV Iintegrase Inhibitors Derived from HIV Gene Products: Structure-Activity Relationship Studies." "Shintaro Suzuki, Kasthuraiah Maddali, Chie Hashimoto, Emiko Urano, Nami Ohashi, Tomohiro Tanaka, Taro Ozaki, Hiroshi Arai, Hiroshi Tsutsumi, Tetsuo Narumi, Wataru Nomura, Naoki Yamamoto, Yves Pommier, Jun A. Komano & Hirokazu Tamamura*" "Bioorg. Med. Chem." 18 6771-6775 2010 10.1016/j.bmc.2010.07.050 原著論文 "Development of Crosslink-Type Tag-Probe Pairs for Fluorescent Imaging of Proteins." "Wataru Nomura, Tomoaki Mino, Tetsuo Narumi, Nami Ohashi, Akemi Masuda, Chie Hashimoto, Hiroshi Tsutsumi & Hirokazu Tamamura*" "Biopolymers: Peptide Science" 94 843-852 2010 10.1002/bip.21444 原著論文 "CD4 Mimics Targeting the Mechanism of HIV entry." "Yuko Yamada, Chihiro Ochiai, Kazuhisa Yoshimura, Tomohiro Tanaka, Nami Ohashi, Tetsuo Narumi, Wataru Nomura, Shigeyoshi Harada, Shuzo Matsushita & Hirokazu Tamamura*" "Bioorg. Med. Chem. Lett." 20 354-358 2010 10.1016/j.bmcl.2009.10.098 原著論文 "Fluorogenically Active Leucine Zipper Peptides as New Tag-Probe Pairs for Protein Imaging in Living Cells." "Hiroshi Tsutsumi, Wataru Nomura, Seiichiro Abe, Tomoaki Mino, Akemi Masuda, Nami Ohashi, Tomohiro Tanaka, Kenji Ohba, Naoki Yamamoto, Kazunari Akiyoshi & Hirokazu Tamamura*" "Angew. Chem., Int. Ed." 48 9164-9166 2009 10.1002/anie.200903183 原著論文 "Structure-activity Relationship Study on Artificial CXCR4 Ligands Possessing the Cyclic Pentapeptide Scaffold: The Exploration of Amino Acid Residues of Pentapeptides by Substitutions of Several Aromatic Amino Acids." "Tomohiro Tanaka, Wataru Nomura*, Tetsuo Narumi, Ai Esaka, Shinya Oishi, Nami Ohashi, Kyoko Itotani, Barry J. Evans, Zi-xuan Wang, Stephen C. Peiper, Nobutaka Fujii & Hirokazu Tamamura*" "Org. Biomol. Chem." 7 3805-3809 2009 10.1039/b908286g 原著論文 "Synthesis of Protein Kinase Cδ C1b Domain by Native Chemical Ligation Methodology and Characterization of Its Folding and Ligand Binding." "Nami Ohashi, Wataru Nomura*, Mai Kato, Tetsuo Narumi, Nancy E. Lewin, Peter M. Blumberg & Hirokazu Tamamura*" "J. Pept. Sci." 15 " 642-646" 2009 10.1002/psc.1161 原著論文 "Structure-activity Relationship Study of CXCR4 Antagonists Bearing the Cyclic Pentapeptide Scaffold: Identification of the New Pharmacophore." "Tomohiro Tanaka, Hiroshi Tsutsumi*, Wataru Nomura, Yasuaki Tanabe, Nami Ohashi, Ai Esaka, Chihiro Ochiai, Jun Sato, Kyoko Itotani, Tsutomu Murakami, Kenji Ohba, Naoki Yamamoto, Nobutaka Fujii & Hirokazu Tamamura*" "Org. Biomol. Chem." 6 "4374-4377 " 2008 原著論文 "Versatile Use of Acid-catalyzed Ring-opening of β-Aziridinyl-α,β-enoates to Stereoselective Synthesis of Peptidomimetics." "Hirokazu Tamamura*, Tomohiro Tanaka, Hiroshi Tsutsumi, Koji Nemoto, Satoko Mizokami, Nami Ohashi, Shinya Oishi & Nobutaka Fujii*" Tetrahedron 63 9243-9254 2007 原著論文 "Multimerized CHR-Derived Peptides as HIV-1 Fusion Inhibitors." "Wataru Nomura, Chie Hashimoto, Takaharu Suzuki, Nami Ohashi, Masayuki Fujino, Tsutoms" "Murakami, Naoki Yamamoto & Hirokazu Tamamura*" "Bioorg. Med. Chem." 21 " 4452-4458 " 2013 10.1016/j.bmc.2013.05.060